Is a
Patent attributes
Patent Jurisdiction
Patent Number
Patent Inventor Names
Giovanna Pescatore0
Caterina Torrisi0
Ester Muraglia0
Philip Jones0
Laura Llauger Bufi0
Olaf Kinzel0
Date of Patent
November 16, 2010
Patent Application Number
12227501
Date Filed
May 29, 2007
Patent Citations Received
Patent Primary Examiner
Patent abstract
The present invention relates to compounds of formula I: and pharmaceutically acceptable salts or tautomers thereof which are inhibitors of poly(ADP-ribose)polymerase (PARP) and thus useful for the treatment of cancer, inflammatory diseases, reperfusion injuries, ischaemic conditions, stroke, renal failure, cardiovascular diseases, vascular diseases other than cardiovascular diseases, diabetes mellitus, neurodegenerative diseases, retroviral infections, retinal damage, skin senescence and UV-induced skin damage, and as chemo- or radiosensitizers for cancer treatment.
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